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Oladapo Bakare

TitleAssociate Professor
Faculty RankAssociate Professor
InstitutionHoward University
DepartmentDepartment of Chemistry
AddressDepartment of Chemistry
Howard University
Washington DC 20059
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    Publications listed below are automatically derived from MEDLINE/PubMed and other sources, which might result in incorrect or missing publications. Faculty can login to make corrections and additions.
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    PMC Citations indicate the number of times the publication was cited by articles in PubMed Central, and the Altmetric score represents citations in news articles and social media. (Note that publications are often cited in additional ways that are not shown here.) Fields are based on how the National Library of Medicine (NLM) classifies the publication's journal and might not represent the specific topic of the publication. Translation tags are based on the publication type and the MeSH terms NLM assigns to the publication. Some publications (especially newer ones and publications not in PubMed) might not yet be assigned Field or Translation tags.) Click a Field or Translation tag to filter the publications.
    1. Akinboye ES, Rosen MD, Bakare O, Denmeade SR. Anticancer activities of emetine prodrugs that are proteolytically activated by the prostate specific antigen (PSA) and evaluation of in vivo toxicity of emetine derivatives. Bioorg Med Chem. 2017 12 15; 25(24):6707-6717. PMID: 29153549.
      Citations:    Fields:    Translation:HumansAnimalsCells
    2. Ogindo CO, Khraiwesh MH, George M, Brandy Y, Brandy N, Gugssa A, Ashraf M, Abbas M, Southerland WM, Lee CM, Bakare O, Fang Y. Novel drug design for Chagas disease via targeting Trypanosoma cruzi tubulin: Homology modeling and binding pocket prediction on Trypanosoma cruzi tubulin polymerization inhibition by naphthoquinone derivatives. Bioorg Med Chem. 2016 08 15; 24(16):3849-55. PMID: 27345756.
      Citations: 3     Fields:    Translation:HumansAnimalsCells
    3. Akinboye ES, Brennen WN, Rosen DM, Bakare O, Denmeade SR. Iterative design of emetine-based prodrug targeting fibroblast activation protein (FAP) and dipeptidyl peptidase IV DPPIV using a tandem enzymatic activation strategy. Prostate. 2016 Jun; 76(8):703-14. PMID: 26835873.
      Citations: 7     Fields:    Translation:HumansCells
    4. Bamji ZD, Washington KN, Akinboye E, Bakare O, Kanaan YM, Copeland RL. Apoptotic Effects of Novel Dithiocarbamate Analogs of Emetine in Prostate Cancer Cell Lines. Anticancer Res. 2015 Sep; 35(9):4723-32. PMID: 26254362.
      Citations: 2     Fields:    Translation:HumansCells
    5. Akinboye ES, Bamji ZD, Kwabi-Addo B, Ejeh D, Copeland RL, Denmeade SR, Bakare O. Design, synthesis and cytotoxicity studies of dithiocarbamate ester derivatives of emetine in prostate cancer cell lines. Bioorg Med Chem. 2015 Sep 01; 23(17):5839-45. PMID: 26187015.
      Citations: 2     Fields:    Translation:HumansCells
    6. Bakare O, Thompson C, Brandy Y, Butcher RJ. 2-Chloro-N-(2-chloro-benzo-yl)-N-(2-ethyl-4-oxo-3,4-di-hydro-quinazolin-3-yl)benzamide. Acta Crystallogr Sect E Struct Rep Online. 2014 Apr 01; 70(Pt 4):o503-4. PMID: 24826190.
    7. Idris N, Butcher RJ, Bakare O. N-(3-Chloro-1,4-dioxo-1,4-di-hydro-naph-thalen-2-yl)-N-propionylpropionamide. Acta Crystallogr Sect E Struct Rep Online. 2014 Feb 01; 70(Pt 2):o102. PMID: 24764835.
    8. Butcher RJ, Berhe S, Anderson AJ, Bakare O. N-Butanoyl-N-(3-chloro-1,4-dioxonaph-thalen-2-yl)butanamide. Acta Crystallogr Sect E Struct Rep Online. 2013; 69(Pt 8):o1230. PMID: 24109321.
    9. Brandy Y, Brandy N, Akinboye E, Lewis M, Mouamba C, Mack S, Butcher RJ, Anderson AJ, Bakare O. Synthesis and characterization of novel unsymmetrical and symmetrical 3-halo- or 3-methoxy-substituted 2-dibenzoylamino-1,4-naphthoquinone derivatives. Molecules. 2013 Feb 04; 18(2):1973-84. PMID: 23381023.
      Citations: 4     Fields:    Translation:Cells
    10. Brandy Y, Butcher RJ, Bakare O. N-(1,4-Dioxo-1,4-dihydro-naphthalen-2-yl)benzamide. Acta Crystallogr Sect E Struct Rep Online. 2012 Sep 01; 68(Pt 9):o2775-6. PMID: 22969654.
    11. Akinboye ES, Rosen MD, Denmeade SR, Kwabi-Addo B, Bakare O. Design, synthesis, and evaluation of pH-dependent hydrolyzable emetine analogues as treatment for prostate cancer. J Med Chem. 2012 Sep 13; 55(17):7450-9. PMID: 22867001.
      Citations: 5     Fields:    Translation:HumansCells
    12. Brandy Y, Butcher RJ, Bakare O. N-Benzoyl-N-(1,4-dioxonaphthalen-2-yl)benzamide. Acta Crystallogr Sect E Struct Rep Online. 2012 Aug 01; 68(Pt 8):o2379. PMID: 22904840.
    13. Ukaegbu M, Butcher RJ, Enwerem NM, Bakare O, Hosten C. 2,3-Dichloro-5,8-dimeth-oxy-1,4-naphtho-quinone. Acta Crystallogr Sect E Struct Rep Online. 2012 Jul 01; 68(Pt 7):o2018. PMID: 22807844.
    14. Khraiwesh MH, Lee CM, Brandy Y, Akinboye ES, Berhe S, Gittens G, Abbas MM, Ampy FR, Ashraf M, Bakare O. Antitrypanosomal activities and cytotoxicity of some novel imido-substituted 1,4-naphthoquinone derivatives. Arch Pharm Res. 2012 Jan; 35(1):27-33. PMID: 22297740.
      Citations: 5     Fields:    Translation:AnimalsCells
    15. Brandy Y, Ononiwu I, Adedeji D, Williams V, Mouamba C, Kanaan Y, Copeland RL, Wright DA, Butcher RJ, Denmeade SR, Bakare O. Synthesis and cytotoxic activities of some 2-arylnaphtho[2,3-d]oxazole-4,9-dione derivatives on androgen-dependent (LNCaP) and androgen-independent (PC3) human prostate cancer cell lines. Invest New Drugs. 2012 Aug; 30(4):1709-14. PMID: 21243402.
      Citations: 4     Fields:    Translation:HumansCells
    16. Kanaan YM, White DF, Das JR, Berhe S, Bakare O, Kenguele H, Beyene D, Zhou Y, Day AA, Copeland RL. Cytotoxic effects of N-(3-chloro-1,4-dioxo 1,4-dihydro-naphthalen-2-yl)-benzamide on androgen-dependent and -independent prostate cancer cell lines. Anticancer Res. 2010 Feb; 30(2):519-27. PMID: 20332464.
      Citations:    Fields:    Translation:HumansCells
    17. Berhe S, Slupe A, Luster C, Charlier HA, Warner DL, Zalkow LH, Burgess EM, Enwerem NM, Bakare O. Synthesis of 3-[(N-carboalkoxy)ethylamino]-indazole-dione derivatives and their biological activities on human liver carbonyl reductase. Bioorg Med Chem. 2010 Jan 01; 18(1):134-41. PMID: 19959367.
      Citations: 2     Fields:    Translation:Humans
    18. Onuegbu J, Butcher RJ, Hosten C, Udeochu UC, Bakare O. Bis(1,10-phenanthroline-5,6-dione-?N,N')silver(I) tetra-fluoridoborate. Acta Crystallogr Sect E Struct Rep Online. 2009 Aug 22; 65(Pt 9):m1119-20. PMID: 21577462.
    19. Akinboye ES, Butcher RJ, Wright DA, Brandy Y, Bakare O. N-(3-Bromo-1,4-dioxo-1,4-dihydro-2-naphth-yl)-4-fluoro-N-(4-fluoro-benzo-yl)benzamide. Acta Crystallogr Sect E Struct Rep Online. 2009 Jan 10; 65(Pt 2):o277. PMID: 21581890.
    20. Kanaan YM, Das JR, Bakare O, Enwerem NM, Berhe S, Beyene D, Williams V, Zhou Y, Copeland RL. Biological evaluation of 2,3-dichloro-5,8-dimethoxy-1,4-naphthoquinone as an anti-breast cancer agent. Anticancer Res. 2009 Jan; 29(1):191-9. PMID: 19331150.
      Citations: 7     Fields:    Translation:HumansCells
    21. Brandy Y, Butcher RJ, Adesiyun TA, Berhe S, Bakare O. 2-Chloro-3-(4-chloro-benzamido)-1,4-naphthoquinone. Acta Crystallogr Sect E Struct Rep Online. 2008 Dec 10; 65(Pt 1):o64. PMID: 21581704.
    22. Akinboye ES, Butcher RJ, Brandy Y, Adesiyun TA, Bakare O. N-(3-Bromo-1,4-dioxo-1,4-dihydro-2-naphth-yl)-2-chloro-N-(2-chloro-benzoyl)benzamide. Acta Crystallogr Sect E Struct Rep Online. 2008 Dec 06; 65(Pt 1):o24. PMID: 21581667.
    23. Singh P, Hallur G, Anchoori RK, Bakare O, Kageyama Y, Khan SR, Isaacs JT. Rational design of novel antiandrogens for neutralizing androgen receptor function in hormone refractory prostate cancer. Prostate. 2008 Oct 01; 68(14):1570-81. PMID: 18668523.
      Citations: 4     Fields:    Translation:HumansCells
    24. Onuegbu J, Butcher RJ, Hosten C, Udeochu UC, Bakare O. 5,6-Di-oxo-1,10-phenanthrolin-1-ium trifluoro-methane-sulfonate. Acta Crystallogr Sect E Struct Rep Online. 2008 Jul 19; 64(Pt 8):o1543. PMID: 21203247.
    25. Onuegbu J, Butcher RJ, Hosten C, Udeochu UC, Bakare O. Acetato(1,10-phenanthroline-5,6-dione)silver(I) trihydrate. Acta Crystallogr Sect E Struct Rep Online. 2008 Jan 25; 64(Pt 2):m403-4. PMID: 21201351.
    26. Copeland RL, Das JR, Bakare O, Enwerem NM, Berhe S, Hillaire K, White D, Beyene D, Kassim OO, Kanaan YM. Cytotoxicity of 2,3-dichloro-5,8-dimethoxy-1,4-naphthoquinone in androgen-dependent and -independent prostate cancer cell lines. Anticancer Res. 2007 May-Jun; 27(3B):1537-46. PMID: 17595773.
      Citations: 8     Fields:    Translation:HumansCells
    27. Udeochu U, Jimerson T, Vivoni A, Bakare O, Hosten CM. Vibrational assignment of the Raman active modes of 1,10-phenanthroline-5,6-dione using DFT calculations. J Phys Chem A. 2007 May 03; 111(17):3409-15. PMID: 17419593.
      Citations: 3     Fields:    
    28. Qiao Z, Udeochu U, Jimerson T, Fletcher M, Bakare O, Hosten CM. Detection of benzopyrene-deoxyguanosine adducts by matrix-assisted laser desorption/ionization time-of-flight mass spectrometry. Rapid Commun Mass Spectrom. 2006; 20(3):487-92. PMID: 16397844.
      Citations:    Fields:    Translation:Cells
    29. Anderson AJ, Nicholson JM, Bakare O, Butcher RJ, Wilson TL, Scott KR. Enaminones 9. Further studies on the anticonvulsant activity and potential type IV phosphodiesterase inhibitory activity of substituted vinylic benzamides. Bioorg Med Chem. 2006 Feb 15; 14(4):997-1006. PMID: 16219468.
      Citations: 2     Fields:    Translation:AnimalsCells
    30. Anderson AJ, Nicholson JM, Bakare O, Butcher RJ, Scott KR. A base-catalyzed solution-phase parallel synthesis of substituted vinylic benzamides from 3-amino-2-cyclohexanones. J Comb Chem. 2004 Nov-Dec; 6(6):950-4. PMID: 15530123.
      Citations: 2     Fields:    Translation:Cells
    31. Bakare O, Ashendel CL, Peng H, Zalkow LH, Burgess EM. Synthesis and MEK1 inhibitory activities of imido-substituted 2-chloro-1,4-naphthoquinones. Bioorg Med Chem. 2003 Jul 17; 11(14):3165-70. PMID: 12818679.
      Citations: 16     Fields:    Translation:HumansCells
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