Evaluation of structural effects on 5-HT(2A) receptor antagonism by aporphines: identification of a new aporphine with 5-HT(2A) antagonist activity.

Ponnala S, Gonzales J, Kapadia N, Navarro HA, Harding WW. Evaluation of structural effects on 5-HT(2A) receptor antagonism by aporphines: identification of a new aporphine with 5-HT(2A) antagonist activity. Bioorg Med Chem Lett. 2014 Apr 01; 24(7):1664-7.

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subject areas

Aporphines
Dose-Response Relationship, Drug
Humans
Molecular Structure
Receptor, Serotonin, 5-HT2A
Structure-Activity Relationship

authors with profiles

Wayne W. Harding

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